High Throughput Screening (HTS): Key issues and the move from research style HTS to industrial style Ultra-High Throughput Screening (UHTS)
(HTS Consulting Ltd.) Jason Armstrong
12:15-14:00
昼食・機器類デモンストレーション
14:00-14:50
Integrated Instrumentation for High Throughput Organic Synthesis
(Charybdis Technologies, Inc.) Thomas J. Baiga
14:50-15:15
Small Molecule Library Synthesis with SynPhaseTM Crowns
(Chiron Technologies Pty. Ltd.) Darryl McConnell
15:15-15:55
Design of New Solid Supports for Combinatorial Chemistry
(Seoul National Univ.) Yoon-Sik Lee
15:55-16:35
Solid and Solution Phase Strategy for the Synthesis of Combinatorial Chemical Libraries
(LG Chemical Ltd.) Sang Woong Kim
16:35-17:25
EVOscreen, a Miniaturized Ultra-High Throughput Screeening System Based on Fluorescence Correlation Spectroscopy (FCS) and Additional Confocal Fluorescence Detection Methods All Having Single-Molecule Sensitivity
(EVOTEC Inc.) Timm Heinrich Jessen
18:00 -
ビア・パーティー
４月２８日（火）
9:30-9:55
進化分子工学による新しいホスト・ゲスト化学の展開
(奈良先端大) 伊藤嘉浩
9:55-10:20
ダイバージェントな経路によるリピドＡ類縁体の合成と生物活性
(阪大・理) ○深瀬嘉之，及川雅人，隅田泰生，深瀬浩一，楠本正一
10:20-10:45
固相 Heck 反応を利用した分子内環化反応
(京都薬科大) 赤路健一
10:45-11:10
デヒドロアラニン誘導体の新規固相合成法
(田辺製薬・医薬拓新研) ○宮島忠利，大野木恵子，岡垣智恵子，山田昌樹
11:10-11:35
チロシン及び両特異性ホスファタ−ゼ阻害活性を持つ低分子ライブラリ−の構築とその構造活性相関
(University of Pittsburgh, 名市大・薬) Robert Rice, James Rusnak, ○横川文明,
横川示帆, Donald Messner, Alton Boynton, Peter Wipf and John Lazo
11:35-12:00
Improving the Efficiency of Lead Optimisation
(BioFocus) Paul Doyle
12:00-12:25
Synthesis and Purification of beta-Amino Alcohol Using "Fish Out" Method
(鐘紡（株）薬品探索研究所化学第１グループ) 堀 学
12:25-14:00
昼休み・機器類デモンストレーション
14:00-14:50
自動合成化学をめざして
(京都大) 吉田潤一
14:50-15:40
Rational Design of Combinatorial Libraries
(MSI) Robert Brown
15:40-16:30
Mass Spectrometric-Based Strategies for Characterizing and Purifyingm Combinatorial Libraries-Developments of a Multi-Column HPLC/MS System
(CombiChem, Inc.) Daniel B. Kassel
16:30-17:20
Biased Secondary Structure Mimetic Libraries for Pharmaceutical Development
