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Japan Combinatorial Chemistry Focus Group

15th Conference on
Combinatorial Chemistry, Japan

On behalf of Japan Combinatorial Chemistry Focus Group, the Organizing Committee cordially invites you to the 15th Conference on Combinatorial Chemistry, Japan (JCCF15).

Sponsored by:	The Japan Combinatorial Chemistry Focus Group
Supported by:	Synthetic Organic Chemistry, Japan
	The Chemical Society of Japan
	The Pharmaceutical Society of Japan

The Conference will emphasize recent major developments in the fields of combinatorial synthesis, robotics synthesis, HTS, and the various related fields.

Transportation to the conference hall

From Tokyo International Airport take the JR train "Narita Express" to JR Tokyo Station (63 min). Take the Marunouchi subway line for Otemachi station (2 min), and change to Hanzomon Line for Chuo-Rinkan via Shibuya. Get off at Mizonokuchi (28 min by express train, 35 min by local train), then take a taxi or free shuttle bus (leave from bus terminal No. 9) for the KSP hotel.

Scientific program

September 18 (Wednesday)
9:30		opening
9:40-10:30	IL-1	Koichi Mikami (Tokyo Institute of Technology) Dynamic Asymmetric Activation: Super High-Throughput Screening of Chiral Ligands and Activators by HPLC-CD/UV and HPLC-OR/RIU
10:30-10:50	O-1	Takayoshi Arai (Osaka University) Diversity and Anisotropy of Complex Molecules
10:50-11:10	O-2	A. D. Baxter,* P. M. Lockey (Argenta Discovery) Hit to "Lead" and "Lead" to "Drug Candidate" Optimisation Using Multi-Parametric Principles
11:10-11:30	O-3	Philipp Ermert, P. Maienfisch, Daniel Obrecht,* T. Pitterna (Polyphor, Ltd) Applications of Sequential Multi-Component Reactions to Focused Libraries
11:30-11:50	O-4	Chikako Saotome,* Osamu Kanie (Mitsubishi Kagaku Institute of Life Sciences) Combinatorial Synthesis of Inhibitors of Glyco-enzymes Based on Induced Fitting
11:50-13:40		Lunch & Exhibition
13:40-14:30	IL-2	Toshihisa Ishikawa (Tokyo Institute of Technology) A New Challenge In The Post-Genome Era: Transport Mechanism-based Drug Design Strategy
14:30-15:20	IL-3	Ferenc Darvas (ComGenex Inc.) Chemical Library Approaches to Target Validation in the Post-Genomic Era
15:20-15:40	O-5	Atsushi Midorikawa (Sumisho Electronics Co., ltd ) Target Library Design by "LeadHopping" using ChemSpace Technology
15:40-16:00	O-6	David E. Patterson,* Richard D. Cramer III (Tripos, Inc.) Improving Purity of Parallel Synthesis Products
16:00-16:20		break
16:20-16:40	O-7	Kiyoshi Nokihara (HiPep Laboratories and Shimadzu Scientific Research Inc.) Construction of a Flexible Synthesis Workstation for Multi-purpose Consisting of Robotic Arm with Different Modules
16:40-17:00	O-8	Hisakazu Mihara1,* Kenji Usui1, Tetsunori Ojima1, Mizuki Takahashi1, Kiyoshi Nokihara2 (1 Dept. of Bioengineering, Tokyo Inst. of Tech., 2 HiPep Laboratories) Peptide Microarrays using Structure-based Libraries for Protein Detection
17:00-17:50	IL-4	John Nielsen (The Royal Veterinary and Agricultural University) Interfacing Natural Product and Combinatorial Chemistry in the Discovery of New Antibiotics
18:00-		Mixer
September 19 (Thursday)
9:00-9:50	IL-5	Kevin Koch (Array BioPharma, Inc.) Developing Superior Human Therapeutics: Exploiting Novel Chemical Genomics Strategies in Drug Discovery
9:50-10:10	O-9	Kosuke Yasuda1,* Steven V. Ley2 (1Tanabe Seiyaku Co., Ltd., 2The University of Cambridge) Oxidations using Solid-Supported Reagents - from Aldehydes and Alcohols to Carboxylic Acids
10:10-10:30	O-10	A. J. Mendonca,* A. F. Coffey, J. W. Davies, F. P. Warner (Polymer Laboratories Inc) Supports for Organic Synthesis: A Comparative Study
10:30-10:50	O-11	Hikaru Takaya,* Shun-Ichi Murahashi (Osaka University) Transition Metal-Based Lewis Acid- and Base-Catalyzed Multicomponent Reactions Directed Toward Combinatorial Chemistry
10:50-11:10	O-12	Takeshi Sagara,* Yufu Sagara, Toshiaki Mase, Toshifumi Kimura, Kazuhito Noguchi, and Norikazu Ohtake (Banyu Pharmaceutical Co., Ltd.) Discovery of a Novel M3 Receptor Selective Antagonist by Combinatorial Chemistry Approach
11:10-12:00	IL-6	Yuichi Hashimoto (Institute of Molecular and Cellular Biosciences, The University of Tokyo) Structural Development of Retinoids and Thalidomide
12:00-13:30		Lunch & Exhibition
13:30-13:50	O-13	Richard Durand (Berger Instruments) Development of an Integrated SFC/MS System to Support Rapid Compound Analysis
13:50-14:10	O-14	Michiko Kanai,* Sachiko Shindo, Masayo Yabu, Michael P. Balogh (Nihon Waters, K.K.) ESCi Multi-mode Ionization Interface for High Throughput LC/MS Analyses of Compound Libraries
14:10-15:00	IL-7	Shuichi Shoji (Waseda University) Recent Trends of Micro Flow Devices and Systems for Chemical/biochemical Applications
15:00-15:20	O-15	Ben Moshiri,* Lewin Wint, Rudy Haidle, Mark Fiskin (Mettler-Toledo AutoChem) Extending the Boundary of Automation: A Solution Phase Synthesizer for Medicinal and Process Chemists
15:20-15:40	O-16	Sergio Romeo (University of Milan, Büchi Labortechnik) Development of a Parallel Synthetic Approach to Ether-Linked Phospholipids Using a Parallel Synthesizer
15:40-16:40	IL-8	Manfred T. Reetz (Max-Planck-Institut für Kohlenforschung) Evolution in the Test Tube as a Means to Create Enantioselective Enzymes

Contributed papers

Contributed papers will be accepted as oral presentations. The organizing committee reserves the right to accept or reject papers. The time for each oral presentation will be 20 or 30 minutes including discussion. Presenters are requested to use OHP or PC projector (35 mm slide projector is not available).
Participants who wish to present a paper should complete Form(RegForm_E.pdf) and send it by FAX to Conference Director of JCCF15 (shown at the bottom of this page) or send following information via e-mail from June 1 to July 16, 2002.


1. Title of paper
   
2. Name(s) of Author(s) (Please mark * for presenting author)
   
3. Affiliation
   
4. e-mail
   

Contributors are requested to supply an abstract by August 8, 2002. Contributors must conform to the Instruction to Contributors(inst_E.pdf).

The conference language, written and spoken will be Japanese and/or English.

Advance registration (by September 10, 2002)
1. associate member: free up to 3 people (An associate member shall pay 100,000 Yen a unit per year. Only associate members can exhibit during the JCCF meetings.)
2. regular member: commercial 15,000 yen; academic, government, public 3,000 yen; student free (A member shall pay 5,000 Yen per year. A student member shall pay 3,000 Yen per year.)
3. member of co-sponsors (e.g., Chemical Society of Japan, Pharmaceutical Society of Japan, etc.): commercial 20,000 yen; academic, government, public 5,000 yen; student 1,000 yen
4. without membership: 30,000 yen
On-site or late registration
1. regular member: commercial 20,000 yen; academic, government, public 5,000 yen; student 1,000 yen.
2. member of co-sponsors: commercial 25,000 yen; academic, government, public 7,000 yen; student 2,000 yen
3. without membership: 40,000 yen

Those who wish to participate in the Conference are kindly requested to register in advance. Please complete Form(RegForm_E.pdf) and send it by FAX to JCCF Society Office (shown at the bottom of this page) or send following information via e-mail from June 1 to September 10, 2002 (for advance registration).


1. Name:
2. Job Title:
3. Organization:
4. Division:
5. Address:
6. City/State/Zip/Country:
7. Phone:
8. Fax:
9. E-mail:

Registration fee must be received prior to the conference.
Payment of the registration fee should be made in Japanese Yen by bank transfer to:

• Name of Bank: Sumitomo Mitsui Bank, Nakanoshimanishi Branch
  
• Account No: (Regular Savings) 3464685
  
• Account Name: Japan Combinatorial Chemistry Focus Group (JCCF)
  

Conference Director


Dr. Takayuki DOI
Department of Appl. Chem., Tokyo Institute of Technology
2-12-1 Ookayama, Meguro, Tokyo 152-8552, Japan
FAX: (+81)-3-5734-2884
E-mail:


Registration


JCCF Society Office
FAX: (+81)-3-3292-7622
E-mail: